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filingDate 2006-03-08-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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publicationDate 2006-09-14-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2006095788-A1
titleOfInvention Particle and preparation containing the particle
abstract Particles of 0.01 to 20 μm average diameter comprising tert-butyl (4R)-4-{[((1R)-2-[(1-benzylpiperidin-4-yl)amino]-1-{[(cyclohexylmethyl)thio]methyl}-2-oxoethyl)amino]carbonyl}-1,3-thiazolidine-3-carboxylate. Preparations comprising the particles excel in transition into the lungs by inhalation and excel in dispersibility as particles, so that handling thereof is easy to thereby enable use of the compound as transpulmonary preparations.
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