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publicationDate 2006-03-30-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2005081960-A3
titleOfInvention Inhibitors of protein tyrosine phosphatase 1b
abstract Protein tyrosine phosphatases (PTPases) such as PTP1B can play a role in regulating a wide variety of cellular responses such as insulin signaling. Substituted bicyclic fused-thiophene compounds can inhibit PTP1B and thereby induce greater insulin sensitivity. Accordingly, PTP1B inhibition can provide an alternate treatment for PTPase-mediated disorders such as diabetes.
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