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filingDate 2004-12-23-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_06c387b5cbe5aa869851c2ff3364ce01
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publicationDate 2005-07-14-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2005062985-A2
titleOfInvention Di-ester prodrugs of camptothecin, process for their preparation and their therapeutical applications
abstract The present invention is related to 10,20-di-O ester derivatives of camptothecin and pharmaceutical formulations thereof. The compounds and pharmaceutical formulations of the present invention possess increased biological life span and bioavailbility and reduced toxicity, while maintaining anti-cancer activity.
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Total number of triples: 746.