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filingDate 2003-07-22-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_f9cfd7beca76025d5ce70bf2771b25c4
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publicationDate 2004-01-29-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-2004010145-A2
titleOfInvention Screening method
abstract A method for identifying test substances that selectively inhibit or activate only a restricted number of transduction pathways of a G-protein-coupled receptor (GPCR) the method comprising the steps of: a) selecting at least one test compound; b) exposing a cell culture, preferably a mammalian cell culture, to the test compound and incubating the culture under suitable conditions; c) selecting at least two distinct intracellular events which are controlled, at least partially, by the G-protein-coupled receptor; d) testing for the ability of said test compound to modulate one of the selected intracellular event; and selecting the test compound which selectively modulates at least one of the pre-selected intracellular event and does not modulate at least another pre­selected intracellular event.
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