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filingDate 2003-05-23-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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publicationDate 2003-12-04-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-03100081-A2
titleOfInvention Biologically active maleamic acid derivatives with labile amide bonds
abstract An process for the reversible modification of membrane interaction of a compound is described. Modification of membrane interaction can be used to facilitate delivery of molecules to cells in vitro and in vivo. The described modifiers, which are used to reversibly inactivate the membrane active compounds, can also be utilized as cross-linkers or to reverse the charge of a molecule.
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Total number of triples: 439.