http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-03084303-A3
Outgoing Links
| Predicate | Object |
|---|---|
| assignee | http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_76ba102ea9c02b6633d64bf09c5b89a4 http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_279273285cf506e06bf39d5aa6a3d953 |
| classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07C311-39 |
| classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07C311-39 |
| filingDate | 2003-03-24-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| inventor | http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_c87ae8ec6ddb12834b627b5e2ed46b19 |
| publicationDate | 2004-08-19-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationNumber | WO-03084303-A3 |
| titleOfInvention | Antagonists of rf-amide neuropeptides |
| abstract | Disclosed are compounds having the formula: (I); where R1 = H, C1-C6 alkyl, cycloalkyl, (a) or (b) (n=1-3); R2 = H, C1-C6 alkyl, cycloalkyl; W= CnH2n-m-NH (n=1-6, m=0, 2, or 4), (c) or (d); X = (e), (f), (g), (h); R3 = (i); Y = (j); Z = CONR8(CH2)n, CONR8(CH2)nCO, P(CH3)OCHR8OCOR9, SO2, SO2(CH2)n, SO2(CH2)nCO, SO2NR8(CH2)n, SO2NR8(CH2)nCO, n=1-4; R4 = H, (CH2)nOH, (CH2)nOCOR10, (CH2)nNR10R11, (CH2)nCONR10R11, n=0-4; R5 = H, (CH2)nNR12R13, N=0-4; R6 = H, (CH2)nNR14R15, n=0-4; R7 = H, C1-C6 alkyl cycloalkyl; R8 = H, C1-C6 alkyl cycloalkyl; R9 = H, C1-C6 alkyl cycloalkyl; R10 = H, C1-C6 alkyl cycloalkyl; R11 = H, C1-C6 alkyl cycloalkyl; R12 = H, C1-C6 alkyl cycloalkyl; R13 = H, C1-C6 alkyl cycloalkyl; R14 = H, C1-C6 alkyl cycloalkyl; R15 = H, C1-C6 alkyl cycloalkyl; Dashed lines: optional; conformational constraint by (CH2)n, n=1-3, R’ =H or O(=) as well as pharmaceuticals compositions and methods for the treatment of opiate addiction, opiate dependence, opiate tolerance, opiate related abstinence syndrome, nicotine addiction and obesity based thereon. |
| priorityDate | 2002-03-29-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| type | http://data.epo.org/linked-data/def/patent/Publication |
Incoming Links
Total number of triples: 16.