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filingDate 2003-02-19-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_7352702775f11f4386ca831990f7b418
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publicationDate 2003-09-04-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-03072033-A2
titleOfInvention Common ligand mimics: thiazolidinediones and rhodanines
abstract The present invention provides common ligand mimics that act as common ligands for a receptor family. The present invention also provides bi-ligands containing these common ligand mimics. Bi-ligands of the invention provide enhanced affinity and/or selectivity of ligand binding to a receptor or receptor family through the synergistic action of the common ligand mimic and specificity ligand which compose the bi-ligand. The present invention also provides combinatorial libraries containing the common ligand mimics and bi-ligands of the invention. Further, the present invention provides methods for manufacturing the common ligand mimics and bi-ligands of the invention and methods for assaying the combinatorial libraries of the invention.
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Total number of triples: 2822.