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filingDate 2003-01-20-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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publicationDate 2003-08-07-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-03064409-A1
titleOfInvention Zoniporide mesylate pharmaceutical compositions and processes for improving solubility of zoniporide
abstract A pharmaceutical composition comprising Zoniporide (N-(5-cyclopropyl-l-quinolin-5yl-lh-pyrazole-4-carbonyl)-guanidine) or its mesylate salt in the presence of an aqueous diluent in the ph range of 2 to 3.5.The composition is a sodium hydrogen exchange-1 (NHE-1)inhibitor for the prevention of,inter alia,perioperative myocardial ischemic injury in mammals.Moreover the application relates to a process for increasing the solubility of Zoniporide employing methanesulfonic acide
priorityDate 2002-01-30-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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