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filingDate 2002-12-04-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_b9343eaf7d49169180c8d3f962033c17
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_bdf3ce65f1c97d30fda8ef715ed6f2dc
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publicationDate 2003-06-12-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-03048127-A1
titleOfInvention Aromatic heterocyclic non-covalent inhibitors of urokinase and blood vessel formation
abstract Novel compounds having activity as non-covalent inhibitors of urokinase and having activity in reducing or inhibiting blood vessel formation are provided. These compounds have at a group having a guanidino moiety or derivative thereof. These compounds are useful in vitro for monitoring plasminogen activator levels and in vivo in treatment of conditions which are ameliorated by inhibition of or decreased activity of urokinase and in treating pathologic conditions wherein blood vessel formation is related to a pathologic condition.
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Total number of triples: 601.