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filingDate 2002-11-29-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_1ff7ce7d4762261500c390995c7cc1b5
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publicationDate 2003-06-05-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-03045913-A1
titleOfInvention Benzamide derivatives, processes for their preparation, and their pharmaceutical use
abstract The present invention relates to novel hydroxyethylene compounds having Asp2 (β-secretase, BACE1 or Memapsin) inhibitory activity, processes for their preparation, to compositions containing them and to their use in the treatment of diseases characterised by elevated β - amyloid levels or β-amyloid deposits, particularly Alzheimer's disease.
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Total number of triples: 571.