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filingDate 2002-08-02-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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publicationDate 2003-02-13-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-03011293-A2
titleOfInvention Pyridinone and pyridazinone derivatives as gonadotropin-releasing hormone receptor antagonists
abstract GnRH receptor antagonists are disclosed having general formula (I), which have utility in the treatment of a variety of sex-hormone related conditions in both men and women. Also disclosed are compositions containing a compound of this invention in combination with a pharmaceutically acceptable carrier, as well as methods relating to the use thereof for antagonizing gonadotropin-releasing hormone in a subject in need thereof.
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Total number of triples: 749.