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classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/G01N33-68
filingDate 2001-09-11-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_ffacb5cead5140a6b13c2cf8c4b00bb6
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_dbb91c199edc3bbc6339670353a93df9
publicationDate 2002-03-14-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-0221135-A2
titleOfInvention Rapid screen to identify p-glycoprotein substrates and high-affinity modulators
abstract A novel method for identifying compounds that interact with P-glycoprotein that involves measuring the quenching of intrinsic tryptophan fluorescence is described. The method has many uses including (1) it can be used to screen drugs for their ability to interact with P-glycoprotein; (2) it can be used to screen for high affinity modulators of P-glycoprotein; and (3) it can be used to screen drugs that are potential hazards when used in combination with the modulators and (4) it can be used in methods of conducting target discovery/screening businesses.
priorityDate 2000-09-11-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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