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filingDate 2001-07-20-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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publicationDate 2002-02-07-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-0210174-A1
titleOfInvention Process for the preparation of 9-amino substituted 9,10-dihydropyrrolo [2,1-b][1,3]benzotiazepines
abstract A process is described for the preparation of compounds with the following formula where the groups are as defined below; in particular, R1 is a substituted amine; said process includes essentially the reaction of pyrrolobenzothiazepin-9-one with amine R1H to give the corresponding enamine, which is subsequently transformed into the final compound.
priorityDate 2000-08-01-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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