http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-02092010-A2

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filingDate 2002-05-16-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_73212753d70c622d6cb92b9315982717
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_77a3a9c849a9282c3c45b96bc62c5329
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publicationDate 2002-11-21-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-02092010-A2
titleOfInvention Reverse-turn mimetics and methods relating thereto
abstract Conformationally constrained compounds which mimic the secondary structure of reverse-turn regions of biologically active peptides and proteins are disclosed. Such compounds have utility over a wide range of fields, including use as diagnostic and therapeutic agents. In particular, compounds of this invention are useful in pharmaceutical compositions as anti-inflammatory agents as well as inhibitors of central nervous disorders. Libraries containing the compounds of this invention are also disclosed, as well as methods for screening the same to identify biologically active members.
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Total number of triples: 498.