Predicate |
Object |
assignee |
http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_5f477632f64551f9c076114eca6a134e http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_3ad907781aeebee3de9f1859911099d0 http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_f5325ab8d0bdd6dc098b2bfbdb29f696 |
classificationCPCInventive |
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D471-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07C251-16 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D209-08 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D209-36 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D207-16 |
classificationIPCInventive |
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D471-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D209-08 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D209-36 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07C251-16 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D207-16 |
filingDate |
2002-03-07-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
inventor |
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_d779a913200b130b0aa88d9fe2fb2c43 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_5017285aaceff8eb69fb8e27bc5ca9a2 |
publicationDate |
2002-09-12-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
publicationNumber |
WO-02070439-A2 |
titleOfInvention |
Amination process |
abstract |
The present invention provides methodology for carbon-nitrogen bond formation via vinyl or aryl amination. In the process of the invention, an sp2 hybridized radical is reacted with an azomethine moiety to form pyrrolidine and indole compounds. The methodology provides a facile process for the synthesis of compounds having the pyrrolidine or indole subunit and is especially advantageous for compounds having acid or base labile functional groups and/or is comprised of chiral centers susceptible to acid/base epimerization. |
priorityDate |
2001-03-07-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
type |
http://data.epo.org/linked-data/def/patent/Publication |