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filingDate 2001-05-17-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_eb9e61b241d8d7ae50db07c7e238a593
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_effa8afb19186e5d597f3e35e89e3a88
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_38bd8246a77aa16e83332f04edf39b59
publicationDate 2001-11-29-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-0190082-A1
titleOfInvention Substituted 1-aminoalkyl-lactams and their use as muscarinic receptor antagonists
abstract This invention relates to compounds which are generally muscarinic M2/M3 receptor antagonists and which are represented by Formula (1) wherein one of X, Y, or Z is independently -S-, -O-, or > N-R4, the others are-CH¿2-;? (p) is an integer from 0 to 3 inclusive; m is an integer from 0 to 3 inclusive; n is an integer from 1 to 6 inclusive; R?3¿ is (C¿1-6?)-alkyl, (C1-6)-alkenyl, (C 1-6)-alkynyl or cycloalkyl; and R?1, R2 and R3¿ are hydrogen or specified substituents. These compounds are useful for treating diseases associated with smooth muscle disorders.
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priorityDate 2000-05-25-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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Total number of triples: 1047.