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filingDate 2001-03-09-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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publicationDate 2001-10-18-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-0177099-A1
titleOfInvention Method for producing benzo annelated heterocycles
abstract A method for producing benzo-annelated heterocycles of general formula (I), wherein X, R<1>, R<2>, R<3>, R<4>, R<5> and n have the meaning cited in Claim 1, by reacting tetrahydrobenzo-annelated heterocycles of formula (II), wherein X, R<1>, R<2>, R<3>, R<4>, R<5>, n and Ac have the meaning cited in Claim 1, with a catalytic amount of an earth metal catalyst in the presence of a hydrodgen acceptor and subsequently deacylating the acylated amino group by adding an amine.
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