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filingDate 2000-10-04-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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publicationDate 2001-04-12-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-0125201-A1
titleOfInvention Process for the preparation of paroxetin intermediate
abstract Compounds of formula (1) where R is an optionally substituted benzyl group, are valuable intermediate in the preparation of paroxetine, and are prepared by reacting a compound of formula (3), where R is as defined for formula (1) with formaldehyde in an acidic medium at elevated temperature.
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