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filingDate 2000-02-11-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_a996e4d310be6c3a69b1b14d42427474
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publicationDate 2001-09-20-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber WO-0047553-A8
titleOfInvention ALKENYL AND ALKYNYL COMPOUNDS AS INHIBITORS OF FACTOR Xa
abstract The invention relates to alkenyl and alkynyl compounds which are potent inhibitors of factor Xa isolated or collected in the prothrombinase complex and to compositions containing said compounds which show a selectivity towards factor Xa greater than that of other proteases. coagulation (e.g. thrombin, fVIIa, fIXa) or fibrinolytic cascades (e.g. plasminogen activators, plasmin). The invention also relates to methods of using said compounds as diagnostic or therapeutic agents for the prevention or treatment in mammals of coagulation disorders such as thromboses.
priorityDate 1999-02-11-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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