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filingDate 2014-03-06-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2018-06-12-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_95f58058ed30c3345a076e0a18c11bf0
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publicationDate 2018-06-12-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-9994525-B2
titleOfInvention H3 antagonists containing phenoxypiperidine core structure
abstract The present invention relates to new histamine H 3 (H 3 ) receptor subtype selective ligands of the general formula (I) and/or geometric isomers and/or stereoisomers and/or diastereomers and/or salts and/or hydrates and/or solvates thereof. The invention further relates to pharmaceutical compositions containing such compounds and the use of these compounds as medicaments for treatment and/or prevention of conditions which require modulation of H 3 receptors. The invention also cover the combinations of a compound of the general formula (I) and an acetylcholinesterase inhibitor.
priorityDate 2013-03-06-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID90389650
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID78705
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID45051774
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID421353896
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID107428
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID23663626
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID16130295
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID90389806
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID90391701
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6251
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID430792788
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID414012638
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID71057243
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID90391703
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226489682
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2332
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID396388
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID405267533
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID90390476
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID4054
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID415897412
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID451180926
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226593861
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID357772
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID118644798
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID447866834
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID118644799
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID430792871
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID118644800
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ867X2
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ867X3
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID11177
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID86298857
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396434
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID86298858
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID458043268
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB4FZ87
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419506070
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID114549
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID466432233
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID86298854
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID681
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID452764334
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID421306191
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP36196
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID86298855
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID58117863
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA0A5G2QVL5
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID9948102
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID86298856
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5202
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226433786
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID452570455
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID405267547
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID448146387

Total number of triples: 353.