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filingDate 2015-09-04-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2017-12-26-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_50b161555302a574ac4d7ceedaa2e8a8
publicationDate 2017-12-26-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-9849138-B2
titleOfInvention 1,4-benzodiazepone-2,5-diones and related compounds with therapeutic properties
abstract The present invention provides novel chemical compounds characterized as Rho kinase (ROCK) inhibitors, methods for their discovery, and their therapeutic, research, and diagnostic use. In particular, the present invention provides 1,4-benzodiazepine-2,5-dione compounds and related compounds having ROCK inhibitory activity, and methods of using such compounds as therapeutic agents to treat a number of conditions associated with ROCK activity.
priorityDate 2009-11-17-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID493931
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226393239
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP81025
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID228304246
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID3085106
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419554365
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID490174
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO93566
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6450551
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226393714
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID3463
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID4543
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID4100
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396220
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226393712
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2008
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419554287
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID282041
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID415728323
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID454216
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID132262553
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396217
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226393698
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID70932979
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396005
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395993
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP81423
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID345512
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395981
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID60916
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226428557
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID157704
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226408986
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID1264
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395967
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5362376
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP07064

Total number of triples: 2873.