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filingDate 2016-11-08-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2017-11-14-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_b688127d941930cb099f7317df02ce8c
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publicationDate 2017-11-14-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-9815805-B2
titleOfInvention Certain (25)-N-[(1S)-1-cyano-2-phenylethyl]-1,4-oxazepane-2-carboxamides as dipeptidyl peptidase 1 inhibitors
abstract The present disclosure relates to certain (2S)-N-[(1S)-1-cyano-2-phenylethyl]-1,4-oxazepane-2-carboxamide compounds (including pharmaceutically acceptable salts thereof), n nthat inhibit dipeptidyl peptidase 1 (DPP1) activity, to their utility in treating and/or preventing clinical conditions including respiratory diseases, such as asthma and chronic obstructive pulmonary disease (COPD), to their use in therapy, to pharmaceutical compositions containing them and to processes for preparing such compounds.
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Total number of triples: 1553.