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filingDate 2016-09-12-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2017-10-17-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_a4b4bb00f3b5d683de2a0e8ab5fac171
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publicationDate 2017-10-17-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-9789199-B2
titleOfInvention MetAP-2 inhibitor polymersomes for therapeutic administration
abstract Described herein are MetAP-2 inhibitors and compositions and formulations thereof, and more particularly compositions and formulations of MetAP-2 inhibitors wherein the MetAP-2 inhibitor is associated with a block copolymer comprising a hydrophilic polymer moiety and a hydrophobic polymer moiety. The present invention also relates to compositions and formulations comprising MetAP-2 inhibitors for oral administration or administration via routes such as topical or ocular administration. The present invention also provides methods to treat conditions associated with or related to the over-expression or over-activity of MetAP-2 by administering the compositions and formulations comprising MetAP-2 inhibitors as disclosed herein.
priorityDate 2007-06-26-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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Total number of triples: 872.