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filingDate 2016-04-27-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2017-09-05-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_5b6692b37698d80b32f18a2e6b5cd3ef
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_9d58cf4a448bbaaac54fddf0efdb5de4
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http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_ab61fe389f9a4747a6fa433412170070
publicationDate 2017-09-05-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-9751858-B2
titleOfInvention 3-heteroaroylamino-propionic acid derivatives and their use as pharmaceuticals
abstract The present invention relates to compounds of the formula I, n nwherein Ht, G, R 10 , R 30 , R 40 , R 50 and R 60 have the meanings indicated in the claims, which are valuable pharmaceutical active compounds. They are inhibitors of the protease cathepsin A, and are useful for the treatment of diseases such as atherosclerosis, heart failure, renal diseases, liver diseases or inflammatory diseases, for example. The invention furthermore relates to processes for the preparation of the compounds of the formula I, their use and pharmaceutical compositions comprising them.
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priorityDate 2011-07-26-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA1JTC4
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA8C8W6
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID425965134
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8A921
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID71269475
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8A9Q8
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ20NV8
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8A341
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8A3I5
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9EA42
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8A4C3
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID71239855
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ0HD57
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396215
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8A1K7
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA5F7A4
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8A1Z5
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5249709
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID424957
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID448420970
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ89YR4
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8A040
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8A061
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID71239829
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID71269442
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA7MN76
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP00723
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID458393758
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA7KGA5
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Total number of triples: 1739.