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filingDate 2014-09-19-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2017-05-23-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_ce2381c835c0d6578e0bcc746eddf8b8
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_7f7d29a6d46638dbcffedf43a50b4232
publicationDate 2017-05-23-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-9656996-B2
titleOfInvention Fused heterocyclic compound, preparation method therefor, pharmaceutical composition, and uses thereof
abstract Disclosed are a fused heterocyclic compound, a preparation method therefor, a pharmaceutical composition, and uses thereof. The preparation method of the fused heterocyclic compound and/or the pharmaceutically acceptable salt thereof in the present invention comprises three synthesizing routes. The present invention also provides a pharmaceutical composition, containing one or more of the fused heterocyclic compound, the pharmaceutically acceptable salt, hydrates, solvent compounds, polymorphs and prodrugs thereof, and a pharmaceutically acceptable carrier. The present invention also relates to an application of the fused heterocyclic compound and/or the pharmaceutical composition in preparing kinase inhibitors and in preparing drugs for preventing and treating diseases related to kinase. The fused heterocyclic compound of the present invention has selective inhibition function on PI3K δ, and can be used for preparing drugs for preventing and treating cell proliferation diseases such as cancers, infections, inflammations, or autoimmune diseases.
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Total number of triples: 891.