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filingDate 2015-03-24-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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publicationDate 2016-12-06-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-9512103-B2
titleOfInvention Synthesis of thiohydantoins
abstract A novel synthesis of the anti-androgen, A52, which has been found to be useful in the treatment of prostate cancer, is provided. A52 as well as structurally related analogs may be prepared via the inventive route. This new synthetic scheme may be used to prepare kilogram scale quantities of pure A52.
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Total number of triples: 1088.