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filingDate 2010-11-01-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2016-11-15-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_b70ae8d6444b523b6097a43347d99522
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publicationDate 2016-11-15-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-9493435-B2
titleOfInvention IRE-1α inhibitors
abstract The invention provides compounds which directly inhibit IRE-1α activity in vitro, prodrugs, and pharmaceutically acceptable salts thereof. Such compounds and prodrugs are useful for treating diseases associated with the unfolded protein response and can be used as single agents or in combination therapies.
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Total number of triples: 2155.