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filingDate 2013-05-09-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2016-05-17-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_9d43e31db7d502f457cb31c9d716878f
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publicationDate 2016-05-17-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-9340537-B2
titleOfInvention Benzamide derivatives for inhibiting the activity of ABL1, ABL2 and BCR-ABL1
abstract The present invention relates to compounds of formula (I): in which Y, Y, R, R 2, R 3 and R 4 are defined in the Summary of the Invention; capable of inhibiting the tyrosine kinase enzymatic activity of the Abelson protein (ABL1), the Abelson-related protein (ABL2) and related chimeric proteins, in particular BCR-ABL1. The invention further provides a process for the preparation of compounds of the invention, pharmaceutical preparations comprising such compounds and methods of using such compounds in the treatment of cancers.
priorityDate 2012-05-15-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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Total number of triples: 2476.