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filingDate 2013-09-09-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2016-05-10-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_5628e4e101e1e0b4c1dfab97e628d5b4
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publicationDate 2016-05-10-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-9334286-B2
titleOfInvention Pharmacologically active compounds
abstract The present invention relates to compounds of formula II n nwherein X, Y, R 2 , R 3 , R 4 and Ar are all as defined herein. The compounds of the present invention are known to inhibit the spindle checkpoint function of Monospindle 1 (Mps1—also known as TTK) kinases either directly or indirectly via interaction with the Mps1 kinase itself. In particular, the present invention relates to the use of these compounds as therapeutic agents for the treatment and/or prevention of proliferative diseases, such as cancer. The present invention also relates to processes for the preparation of these compounds, and to pharmaceutical compositions comprising them.
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID428531773
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP51744
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID451897553
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID428531776
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID89995584
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID227039654
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID223746476
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID413823327
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ6YK33
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP51748
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID311716646
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID73389263
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ6YRB1
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID422228477
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ15797
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCF1N1G1
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID138223
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ71WN4
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID89995583
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID311716660
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP12708
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID89995592
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Total number of triples: 2737.