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inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_3732a2b5d0c0f6451d6a7baba5c75a37
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publicationDate 2016-04-26-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-9321743-B2
titleOfInvention Compositions and methods of inhibiting N-acylethanolamine-hydrolyzing acid amidase
abstract Compounds and pharmaceutical compositions are contemplated that inhibit N-acyl-ethanolamine-hydrolyzing acid amidase (NAAA) to so increase the concentration of the substrate of NAAA, palmitoylethanolamide (PEA). NAAA inhibition is contemplated to be effective to alleviate conditions associated with a reduced concentration of PEA. Among other uses, various NAAA inhibitors are especially contemplated as therapeutic agents in the treatment of inflammatory diseases.
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