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filingDate 2012-03-31-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2016-03-22-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_0cfac6c7eeb070a6ecc6e69ca472a6a1
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publicationDate 2016-03-22-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-9290460-B2
titleOfInvention 1-(Arylmethyl)quinazoline-2,4(1H,3H)-diones as PARP inhibitors and the use thereof
abstract Disclosed are 1-(arylmethyl)quinazoline-2,4(1H,3H)-diones thereof, represented by the Formula (I) wherein Ar, R 1 -R 6 are defined herein. Compounds having Formula (I) are PARP inhibitors. Therefore, compounds of the invention may be used to treat clinical conditions that are responsive to the inhibition of PARP activity.
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Total number of triples: 1122.