http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-9216986-B1

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filingDate 2012-12-21-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2015-12-22-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_f47aa5644e0bbef016ea62866a714e14
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_1dd35e181f0efb66952b49bb7b31d43a
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publicationDate 2015-12-22-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-9216986-B1
titleOfInvention Quinoline derivatives as PDE10A enzyme inhibitors
abstract The present invention provides quinoline derivatives of formula I that are PDE10A enzyme inhibitors, and as such are useful to treat neurodegenerative and psychiatric disorders. Especially, the invention provides compounds that are highly selective for PDE10 over other PDE subtypes. The present invention also provides pharmaceutical compositions comprising compounds of the invention and methods of treating disorders using the compounds of the invention.
priorityDate 2011-12-21-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP01328
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID395564
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ86C56
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226572306
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID431833584
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP01330
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID154073757
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ29450
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP9WMU8
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ91WF3
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID118588257
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID458393376
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID154073758
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP01321
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID227101248
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP9WMU9
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP01324
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID89649658
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID127552948
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226572305
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID118588255
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID431833553
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP01319
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID431173888
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID318488886
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID978
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID318488885
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID89650369
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID433015734
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID431173897
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP01320
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP01316
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID431173844
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID118588254
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID451465078
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP01317
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID431173853
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID7060
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID7745
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID160054548
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID318488871
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID318488872
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP01342
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ09435
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID118588269

Total number of triples: 985.