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filingDate 2010-12-22-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2015-12-22-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_383ad8ffd927753e696cf5d0579dfc5e
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_a74024b40b18f6308fcde817bedec886
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publicationDate 2015-12-22-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-9216975-B2
titleOfInvention TRPV1 vanilloid receptor antagonists with a bicyclic portion
abstract The invention discloses compounds of formula I n n n n n n n n n n n n wherein Y is a group of formula A, B, C, D, or E: n n n n n n n n n n n n n n n n and W, Q, n, R1, R2, R3, U1-U5, J and K have the meanings given in the description. n n n n n The compounds of formula I are TRPV1 antagonists and are useful as active ingredients of pharmaceutical compositions for the treatment of pain and other conditions ameliorated by the inhibition of the vanilloid receptor TRPV1.
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priorityDate 2010-03-30-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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Total number of triples: 1087.