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filingDate 2014-01-10-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2015-08-18-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_292e74ba01b5651f516b54748eaa27b3
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publicationDate 2015-08-18-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-9108955-B2
titleOfInvention Heterocyclic inhibitors of necroptosis
abstract The invention features a series of heterocyclic derivatives that inhibit tumor necrosis factor alpha (TNF-α) induced necroptosis. The heterocyclic compounds of the invention are described by Formulas (I) and (Ia)-(Ie) and are shown to inhibit TNF-α induced necroptosis in FADD-deficient variant of human Jurkat T cells. The invention further features pharmaceutical compositions featuring the compounds of the invention. The compounds and compositions of the invention may also be used to treat disorders where necroptosis is likely to play a substantial role.
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID324199100
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID25190402
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID327563205
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID453409477
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID25190405
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID85854492
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID325873097
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2773578
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID25190404
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID25189824
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID323035074
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226397462
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID16249
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID53394777
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395155
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID25190406
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226397531
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID637517
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID248747247
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID7505
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID425520775
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID146921336
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID7504
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID228304246
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID70790375
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226394128
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID71100778
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID161057133
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID24755357
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID98564
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID3893
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID8420
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID425676690
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID162229893
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID237874703
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID24857830
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID237874678
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID325878560
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395968

Total number of triples: 644.