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filingDate 2011-02-25-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2015-03-03-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_5cdb9ed88f3283e953eb76fde69b841a
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publicationDate 2015-03-03-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-8969376-B2
titleOfInvention Pyrazolopyrimidine compounds and their use as PDE10 inhibitors
abstract The present invention relates to a compound represented by formula [I]: n nwherein:n R 1 is hydrogen, halogen, lower alkyl or cyano; Ring A is an optionally substituted heterocyclic group; Ring B is an optionally substituted 3 to 6-membered monocyclic group; and Y is optionally substituted amino, optionally substituted cyclic amino, optionally substituted aliphatic 3 to 6-membered monocyclyloxy, optionally substituted lower alkyl or optionally substituted lower alkyl-O—,n nor a pharmaceutically acceptable salt thereof, and to their use as PDE10 inhibitor.
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Total number of triples: 2758.