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filingDate 2010-10-13-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2014-09-30-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_8573e0dc59e3e8cc9455ea68714ea5cd
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publicationDate 2014-09-30-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-8846110-B2
titleOfInvention Polymeric systems for the delivery of anticancer drugs
abstract The present invention relates to compositions for the treatment of cancerous tissues in warm-blooded animals containing one or two anticancer agents attached to polymeric carriers having monomer units derived from one or more of N-(2-carboxypropyl)methacrylamide (2-CPMA), N-(3-carboxypropyl)methacrylamide (3-CPMA), N-(2-aminopropyl)methacrylamide (2-APMA) and/or N-(3-aminopropyl)methacrylamide (3-APMA) are also included. Anticancer agents in compositions can be attached to said polymeric carrier by side-chains which can be susceptible to hydrolysis by lysosomal enzymes intracellularly. Compositions can also include a targeting ligand attached to the polymeric carrier, optionally through a second linker.
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