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publicationDate 2014-08-26-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-8815908-B2
titleOfInvention Compounds and methods for inhibiting phosphate transport
abstract Compounds having activity as phosphate transport inhibitors, more specifically, inhibitors of intestinal apical membrane Na/phosphate co-transport, are disclosed. The compounds have the following structure (I): n nincluding stereoisomers, pharmaceutically acceptable salts and prodrugs thereof, wherein X, Y, R 1 and R 2 are as defined herein. Methods associated with preparation and use of such compounds, as well as pharmaceutical compositions comprising such compounds, are also disclosed.
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Total number of triples: 506.