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filingDate 2009-12-16-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2014-06-17-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_f90ca24ce40489affa38e303dfdf7bbe
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publicationDate 2014-06-17-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-8754261-B2
titleOfInvention Process for the preparation of O-desmethyl-venlafaxine and salts thereof
abstract The present invention relates to a novel process for the preparation of O-desmethyl venlafaxine (ODV) and the pharmaceutically acceptable salts thereof, wherein it comprises (i) provision of spiro-venlafaxine compound as intermediate; (ii) conversion of spiro-venlafaxine intermediate into ODV free base in a one-pot process; and (iii) optionally conversion ODV free base into pharmaceutically acceptable salts. The present invention further relates to novel processes for the preparation of crystalline salts of ODV-succinate and ODV-oxalate.
priorityDate 2009-12-16-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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