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publicationDate 2014-06-10-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-8748418-B2
titleOfInvention 1,4-oxazepines as BACE1 and/or BACE2 inhibitors
abstract The present invention relates to 1,4-Oxazepines of formula I n nhaving BACE1 and/or BACE2 inhibitory activity, their manufacture, pharmaceutical compositions containing them and their use as therapeutically active substances. The active compounds of the present invention are useful in the therapeutic and/or prophylactic treatment of e.g. Alzheimer's disease and type 2 diabetes.
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Total number of triples: 1967.