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publicationDate 2014-06-10-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-8748415-B2
titleOfInvention C-28 amines of C-3 modified betulinic acid derivatives as HIV maturation inhibitors
abstract Compounds having drug and bio-affecting properties, their pharmaceutical compositions and methods of use are set forth. In particular, C-28 amines of C-3 modified betulinic acid derivatives that possess unique antiviral activity are provided as HIV maturation inhibitors. These compounds are useful for the treatment of HIV and AIDS. In particular, the following compounds are provided herein, including pharmaceutically acceptable salts thereof: n a compound of formula I n na compound of formula IIn n nand a compound of formula III
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Total number of triples: 3018.