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filingDate 2011-06-06-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2014-05-13-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_d0e1ec3f6e2864ec0ff6b11b8ba37313
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publicationDate 2014-05-13-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-8722629-B2
titleOfInvention Auristatin derivatives and use thereof
abstract The present application relates to novel derivatives of monomethylauristatin F, to processes for preparing these derivatives, to the use of these derivatives for treating and/or preventing diseases, and also to the use of these derivatives for preparing medicaments for treating and/or preventing diseases, more particularly hyperproliferative and/or angiogenic disorders such as, for example, cancerous disorders. Such treatments may be practised as a monotherapy or else in combination with other medicaments or further therapeutic measures.
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Total number of triples: 1359.