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filingDate 2010-07-26-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2014-03-25-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_721f6a0e76ddaaa468c15337817a5887
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publicationDate 2014-03-25-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-8680120-B2
titleOfInvention Indole derivative or pharmaceutically acceptable salt thereof
abstract A compound (I) of the present invention, which has an EP 1 receptor antagonism: n n n n n n n n n n n n [wherein A represents a benzene ring or the like; Y 1 represents a C 1-6 alkylene group; Y 2 represents a single bond or the like; R 1 represents a hydrogen atom, a C 1-6 alkyl group or the like; R 2 represents a phenyl group which may have a substituent, a 5-membered aromatic heterocyclic ring which may have a substituent, a 6-membered aromatic heterocyclic ring which may have a substituent or the like; R 3 represents a halogen atom, a C 1-6 alkoxy group or the like; R 4 represents a hydrogen atom or the like; and R 5 represents a hydrogen atom or the like] or a pharmaceutically acceptable salt thereof is provided. Furthermore, the compound (I) of the present invention can be used as an agent for treating or preventing LUTS, in particular, various symptoms of OABs.
priorityDate 2009-07-27-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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Total number of triples: 2922.