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filingDate 2010-12-09-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2014-03-04-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_1c1d4ed62955d08e5dcfac657be6d0f3
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publicationDate 2014-03-04-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-8664387-B2
titleOfInvention Pyridoquinazolinone M1 receptor positive allosteric modulators
abstract The present invention is directed to quinolinone-pyrazolone compounds of formula (I) which are M1 receptor positive allosteric modulators and that are useful in the treatment of diseases in which the M1 receptor is involved, such as Alzheimer's disease, schizophrenia, pain or sleep disorders. The invention is also directed to pharmaceutical compositions comprising the compounds, and to the use of the compounds and compositions in the treatment of diseases mediated by the M1 receptor.
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type http://data.epo.org/linked-data/def/patent/Publication

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Total number of triples: 1787.