http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-8580813-B2

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classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-44
filingDate 2010-07-28-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2013-11-12-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_799f7e3ff386bbbd71f16440606ef1d6
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_03df9b04670c90fce8ca89f215bb59cb
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publicationDate 2013-11-12-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-8580813-B2
titleOfInvention Cyclic azaindole-3-carboxamides, their preparation and their use as pharmaceuticals
abstract The present invention relates to cyclic azaindole-3-carboxamides of the formula I, n nwherein A, R, R 10 , R 20 , R 30 , R 40 , Y 1 , Y 2 , Y 3 , Y 4 , n, p and q have the meanings indicated in the claims, which are valuable pharmaceutical active compounds. Specifically, they inhibit the enzyme renin and modulate the activity of the renin-angiotensin system, and are useful for the treatment of diseases such as hypertension, for example. The invention furthermore relates to processes for the preparation of the compounds of the formula I, their use and pharmaceutical compositions comprising them.
priorityDate 2008-01-31-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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Total number of triples: 2086.