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filingDate 2010-09-03-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2013-11-12-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_eece9eaf2c65fb00b81f6fddd7531eb4
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publicationDate 2013-11-12-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-8580783-B2
titleOfInvention [1,2,4]triazolo [1,5-c]pyrimidine derivatives as Hsp90 modulators
abstract The present invention relates to [1,2,4]triazolo[1,5-c]pyrimidine derivatives of formula (I) which inhibit the activity of Heat Shock Protein Hsp90. The compounds of the invention are therefore useful in treating proliferative diseases such as cancer and neurodegenerative diseases. The present invention also provides processes for preparing these compounds, methods of treating diseases and the pharmaceutical compositions comprising these compounds.
priorityDate 2009-09-10-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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Total number of triples: 1856.