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classificationCPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D471-04
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classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-44
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D221-22
filingDate 2011-06-10-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2013-10-15-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_320b7516cc10feca46c08ec6dcf38627
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_76f3ba5d0a7df941656b912652c8443f
publicationDate 2013-10-15-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-8557992-B2
titleOfInvention Heterocyclic fused phenanthrolinone M1 receptor positive allosteric modulators
abstract The present invention is directed to heterocyclic fused phenanthrolinone compounds of formula (I) which are M1 receptor positive allosteric modulators and that are useful in the treatment of diseases in which the M1 receptor is involved, such as Alzheimer's disease, schizophrenia, pain or sleep disorders. The invention is also directed to pharmaceutical compositions comprising the compounds, and to the use of the compounds and compositions in the treatment of diseases mediated by the M1 receptor.
isCitedBy http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-2023114224-A1
priorityDate 2010-06-15-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID129514880
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5460631
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID746942
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Total number of triples: 1640.