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filingDate 2008-08-04-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2013-08-27-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_6944e9c662519a79f7fd46d1b50804b7
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publicationDate 2013-08-27-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-8518916-B2
titleOfInvention Heterocyclic derivatives as M-GLU5 antagonists
abstract This invention relates to novel heterocyclic compounds having selective affinity for the mGlu5 subtype of metabotropic receptors, pharmaceutical compositions thereof and uses for such compounds and compositions in the treatment of lower urinary tract disorders, such as neuromuscular dysfunction of the lower urinary tract, and in the treatment of migraine and gastroesophagael reflux disease (GERD).
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Total number of triples: 4218.