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filingDate 2009-08-05-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2013-07-16-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_ad1f71d8c96b63083f4bbddea90fa61a
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publicationDate 2013-07-16-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-8486964-B2
titleOfInvention Fused pyrrolidino-cyclopropane derivatives as selective 11-beta-hydroxysteroid dehydrogenase type 1 inhibitors
abstract The present invention relates to fused pyrrolidino-cyclopropane derivatives according to formulae (I) to (IV) as selective inhibitors of the enzyme 11-beta-hydroxysteroid dehydrogenase type 1 (11-β-HSD-1) and the use of such compounds for the treatment and/or prevention of metabolic syndrome, diabetes, insulin resistance, obesity, lipid disorders, glaucoma, osteoporosis, cognitive disorders, anxiety, depression, immune disorders, hypertension and other diseases and conditions.
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID568
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID16051939
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID444254
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6385
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226479487
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID439260
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID244004515
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID453
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396738
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID53690099
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226397660
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID128334896
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5541
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID160869790
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID41214
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226393254
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID12766
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID760
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID31257
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5798
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID322897900
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226393239
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID129559307
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID223752024
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID17774203
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID80005
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226407215
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID8125
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID128279931
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID985
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID12350

Total number of triples: 647.