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publicationDate 2013-04-09-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-8415367-B2
titleOfInvention Pyrimidinylpiperidinyloxypyridinone analogues as GPR119 modulators
abstract Novel compounds of structure Formula I: n nor an enantiomer, a diastereomer, or a pharmaceutically acceptable salt thereof, wherein n 1 , R 1 , R 2 , R 3 and R 4 are defined herein, are provided which are GPR119 G protein-coupled receptor modulators. GPR119 G protein-coupled receptor modulators are useful in treating, preventing, or slowing the progression of diseases requiring GPR119 G protein-coupled receptor modulator therapy. Thus, the disclosure also concerns compositions comprising these novel compounds and methods of treating diseases or conditions related to the activity of the GPR119 G protein-coupled receptor by using any of these novel compounds or a composition comprising any of such novel compounds.
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Total number of triples: 2172.