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publicationDate 2013-01-22-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-8357506-B2
titleOfInvention Method of identifying improved conjugates of biologically active compounds
abstract This invention features a method of identifying a compound useful for enhancing efficacy of a therapeutic agent. The method includes incubating a compound in blood cells; separating immune cells from erythrocytic cells; and determining the ratio of the concentration of the compound in the immune cells to the concentration of the compound in the erythrocytic cells; wherein the compound comprises a transportophore and a therapeutic agent, in which the transportophore is covalently bonded to the therapeutic agent via a bond or a linker.
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Total number of triples: 1482.